Product name: PK20
Synonyms: opioid-neurotensin hybrid peptide PK20,
Sequence: Dmt-D-Lys-Phe-Phe-Lys-Lys-Pro-Phe-Tle-Leu-OH
Purity: 95% by HPLC
Counter ion: Trifluoacetate
Format: Lyophilized powder
Description: A novel compound (PK20, Dmt-D-Lys-Phe-Phe-Lys-Lys-Pro-Phe-Tle-Leu-OH) targets single entity opioid and neurotensin pharmacophores. This endomorphin-2-like opioid peptide was introduced as a highly active analgesic because it elicited a strong dose- and time-dependent antinociceptive response when administered centrally and peripherally. Its pain-relieving activity was observed as rapidly as 5 min after drug injection.
Usage: For Scientific Research Use Only, Not for Human Use.
Reference:
European Journal of Pharmaceutical Sciences, Volume 63, 15 October 2014, Pages 8-13.
Pharmacological Reports.Volume 65, Issue 4, July–August 2013, Pages 836–846.